In the world of Tracazolate, there are endless aspects to discover and explore. From its origins to its relevance today, Tracazolate has captured the attention of millions of people around the world. Whether through its influence on popular culture, its impact on society or its importance in times past, Tracazolate continues to spark interest and generate debate. In this article, we will delve into the fascinating world of Tracazolate, exploring its different facets and unraveling its meaning in the current context. From its evolution over the years to its role in people's lives, Tracazolate is a topic that deserves to be analyzed from various perspectives to understand its true magnitude.
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Routes of administration | By mouth |
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ECHA InfoCard | 100.050.178 |
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Formula | C16H24N4O2 |
Molar mass | 304.394 g·mol−1 |
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Tracazolate (ICI-136,753) is an anxiolytic drug which is used in scientific research. It is a pyrazolopyridine derivative, most closely related to pyrazolopyrimidine drugs such as zaleplon, and is one of a structurally diverse group of drugs known as the nonbenzodiazepines which act at the same receptor targets as benzodiazepines but have distinct chemical structures.
Tracazolate has primarily anxiolytic and anticonvulsant effects, with sedative and muscle relaxant effects only appearing at higher doses. It has a unique receptor binding profile involving allosteric modulation of several GABAA receptor subtypes, being selective for GABAA receptors containing α1 and β3 subunits, but exhibiting different effects depending on the third type of subunit making up the receptor complex.